Octanoic acid ( CPI-613 )

产品货号. M16844 CAS No. 95809-78-2

COA

Datasheet

HNMR

HPLC

MSDS

Handing Instructions

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产品名称

Octanoic acid
注意事项

本公司产品仅用于科研实验，不得用于人体或动物的临床与诊断
产品简述

CPI-613, a lipoate analog, inhibits mitochondrial enzymes pyruvate dehydrogenase (PDH) and α-ketoglutarate dehydrogenase, disrupts tumor cell mitochondrial metabolism.
产品描述

CPI-613, a lipoate analog, inhibits mitochondrial enzymes pyruvate dehydrogenase (PDH) and α-ketoglutarate dehydrogenase, disrupts tumor cell mitochondrial metabolism. Phase 2.
同义词

CPI-613
通路

Metabolic Enzyme/Protease
靶点

Dehydrogenase
受体

α-ketoglutarate dehydrogenase; PDH
研究领域

Cancer
适应症

——

CAS Number

95809-78-2
分子量

388.59
分子式

C22H28O2S2
纯度

>98%(HPLC)
溶解度

DMSO:78 mg/mL (200.72 mM); Ethanol:78 mg/mL (200.72 mM); Water:<1 mg/mL (<1 mM)
SMILES

O=C(O)CCCCC(SCC1=CC=CC=C1)CCSCC2=CC=CC=C2
化学全称

6,8-bis(benzylthio)octanoic acid

1. Zachar Z, et al. J Mol Med (Berl). 2011, 89(11), 1137-1148.

计算器

产品手册

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